*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : SO2519500
CHEMICAL NAME : 10H-Phenothiazine,
2-chloro-10-(3-(3-methyl-3,9-diazabicyclo(3.3.1)non-9
-yl)propyl)-, dihydrochloride
CAS REGISTRY NUMBER : 27447-78-5
LAST UPDATED : 198209
DATA ITEMS CITED : 2
MOLECULAR FORMULA : C23-H28-Cl-N3-S.2Cl-H
MOLECULAR WEIGHT : 486.97
WISWESSER LINE NOTATION : T C666 BN ISJ EG B3- AT66 A AN DNTJ D1 &GH 2
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* 2-Chloro-10-(3-(3-methyl-3,9-diazabicyclo(3.3.1)non-9-yl)propyl)-10H-phe
nothiazine 2HCl
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intraperitoneal
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 155 mg/kg
TOXIC EFFECTS :
Behavioral - antipsychotic
REFERENCE :
RPTOAN Russian Pharmacology and Toxicology (English Translation).
Translation of FATOAO. (Euromed Pub., 33, Woodlands Rd., Surbiton, Surrey,
UK) V.30- 1967- Volume(issue)/page/year: 35,162,1972
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intravenous
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 93 mg/kg
TOXIC EFFECTS :
Behavioral - rigidity (including catalepsy)
REFERENCE :
RPTOAN Russian Pharmacology and Toxicology (English Translation).
Translation of FATOAO. (Euromed Pub., 33, Woodlands Rd., Surbiton, Surrey,
UK) V.30- 1967- Volume(issue)/page/year: 35,162,1972
*** END OF RECORD ***