*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : KE2100000
CHEMICAL NAME : Ergoline-8-beta-carboxamide,
1-acetyl-9,10-didehydro-N,N-diethyl-6-methyl-,
bitartrate
CAS REGISTRY NUMBER : 63938-24-9
LAST UPDATED : 199012
DATA ITEMS CITED : 2
MOLECULAR FORMULA : C22-H27-N3-O2.2C4-H4-O6
MOLECULAR WEIGHT : 661.68
WISWESSER LINE NOTATION : T C6656 1A P GN LN CUTT&&J EVN1&1 G1 LV1 &OVYQYQVO 2
COMPOUND DESCRIPTOR : Human
SYNONYMS/TRADE NAMES :
* 1-Acetyl-9,10-didehydro-N,N-diethyl-6-methylergoline-8-beta-carboxamide
bitartrate
* 1-Acetyllysergic acid diethylamide bitartrate
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE : Oral
SPECIES OBSERVED : Human
DOSE/DURATION : 1500 ng/kg
TOXIC EFFECTS :
Brain and Coverings - changes in surface EEG
Behavioral - hallucinations, distorted perceptions
Behavioral - changes in psychophysiological tests
REFERENCE :
PSDTAP Proceedings of the European Society for the Study of Drug Toxicity.
(Princeton, NJ 08540) V.1-15, 1963-74. For publisher information, see
PESTD5. Volume(issue)/page/year: 8,59,1967
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intravenous
SPECIES OBSERVED : Rodent - rabbit
DOSE/DURATION : 1600 ug/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
27ZQAG "Psychotropic Drugs and Related Compounds," 2nd ed., Usdin, E., and
D.H. Efron, Washington, DC, 1972 Volume(issue)/page/year: -,93,1972
*** END OF RECORD ***