*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : HP5295000
CHEMICAL NAME : Dibenzofuran, 3-methoxy-4-pyrrolidinomethyl-
CAS REGISTRY NUMBER : 42840-17-5
LAST UPDATED : 199012
DATA ITEMS CITED : 4
MOLECULAR FORMULA : C18-H19-N-O2
MOLECULAR WEIGHT : 281.38
WISWESSER LINE NOTATION : T B656 HOJ EO1 F1- AT5NTJ
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* 3-Methoxy-4-pyrrolidinylmethyldibenzofuran
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Oral
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 838 mg/kg
TOXIC EFFECTS :
Behavioral - excitement
REFERENCE :
TAKHAA Takeda Kenkyusho Ho. Journal of the Takeda Research Laboratories.
(Takeda Yakuhin Kogyo K.K., 2-17-85 Jusohon-machi, Yodogawa-ku, Osaka 532,
Japan) V.29- 1970- Volume(issue)/page/year: 31,247,1972
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intraperitoneal
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 90 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
CHTPBA Chimica Therapeutica. (Paris, France) V.1-8, 1965-73. For
publisher information, see EJMCA5. Volume(issue)/page/year: 8,57,1973
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Oral
SPECIES OBSERVED : Primate - monkey
DOSE/DURATION : 1000 ug/kg
TOXIC EFFECTS :
Blood - aplastic anemia
Nutritional and Gross Metabolic - weight loss or decreased weight gain
Biochemical - Metabolism (Intermediary) - other
REFERENCE :
ANYAA9 Annals of the New York Academy of Sciences. (New York Academy of
Sciences, 2 E. 63rd St., New York, NY 10021) V.1- 1877-
Volume(issue)/page/year: 320,151,1979
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Oral
SPECIES OBSERVED : Rodent - guinea pig
DOSE/DURATION : 10 ug/kg
TOXIC EFFECTS :
Behavioral - withdrawal
Skin and Appendages - hair
Nutritional and Gross Metabolic - weight loss or decreased weight gain
REFERENCE :
ANYAA9 Annals of the New York Academy of Sciences. (New York Academy of
Sciences, 2 E. 63rd St., New York, NY 10021) V.1- 1877-
Volume(issue)/page/year: 320,151,1979
*** END OF RECORD ***