*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : CV2369000
CHEMICAL NAME : Benzamide,
3-bromo-2,6-dimethoxy-N-(1-ethyl-2-pyrrolidinylmethyl
)-, hydrochloride, (S)-(-)-
CAS REGISTRY NUMBER : 73220-03-8
LAST UPDATED : 199412
DATA ITEMS CITED : 1
MOLECULAR FORMULA : C16-H23-Br-N2-O3
MOLECULAR WEIGHT : 371.32
WISWESSER LINE NOTATION : T5NTJ A2 B1MVR CE BO1 FO1 &GH
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* (S)-(-)-2-((3-Bromo-2,6-dimethoxybenzamido)methyl)-1-ethylpyrrolidine
hydrochloride
* (S)-(-)-3-Bromo-2,6-dimethoxy-N-(1-ethyl-2-pyrrolidinylmethyl)benzamide
hydrochloride
* (-)-Fla 732
* Remoxipride hydrochloride
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intraperitoneal
SPECIES OBSERVED : Rodent - rat
DOSE/DURATION : 324 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity)
Behavioral - rigidity (including catalepsy)
REFERENCE :
JMCMAR Journal of Medicinal Chemistry. (American Chemical Soc.,
Distribution Office Dept. 223, POB POB 57136, West End Stn., Washington, DC
20037) V.6- 1963- Volume(issue)/page/year: 25,1280,1982
*** END OF RECORD ***