*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : CF2080000
CHEMICAL NAME : L-Arginine, N(sup
2)-(N-(N-(N-(L-tyrosyl-D-alanyl)glycyl)-L-phenylalany
l)-L-leucyl)-
CAS REGISTRY NUMBER : 81733-79-1
BEILSTEIN REFERENCE NO. : 4287455
LAST UPDATED : 199612
DATA ITEMS CITED : 2
MOLECULAR FORMULA : C35-H51-N9-O8
MOLECULAR WEIGHT : 725.95
SYNONYMS/TRADE NAMES :
* Dalargin
* Tyrosyl-D-alanyl-glycyl-phenylalanyl-leucyl-arginine
* N(sup
2)-(N-(N-(N-(L-Tyrosyl-D-alanyl)glycyl)-L-phenylalanyl)-L-leucyl)-L-argi
nine
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intravenous
SPECIES OBSERVED : Rodent - rat
DOSE/DURATION : 270 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
DRFUD4 Drugs of the Future. (J.R. Prous, S.A., Apartado de Correos 540,
08080 Barcelona, Spain) V.1- 1975/76- Volume(issue)/page/year:
16,203,1991
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intravenous
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 520 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
DRFUD4 Drugs of the Future. (J.R. Prous, S.A., Apartado de Correos 540,
08080 Barcelona, Spain) V.1- 1975/76- Volume(issue)/page/year:
16,203,1991
*** END OF RECORD ***