*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : UX9712000
CHEMICAL NAME : Pyrrolidine, 1-benzyl-2,5-bis(chloromethyl)-,
hydrochloride
LAST UPDATED : 199506
DATA ITEMS CITED : 3
MOLECULAR FORMULA : C13-H17-Cl2-N.Cl-H
MOLECULAR WEIGHT : 294.67
WISWESSER LINE NOTATION : T5NTJ A1R& B1G E1G
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* N-Benzil-2,5-bis-(clorometil)-pirrolidina cloridrato
* 1-Benzyl-2,5-bis(chloromethyl)pyrrolidine hydrochloride
* ERL-491
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Oral
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 500 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
JMPCAS Journal of Medicinal and Pharmaceutical Chemistry. (Washington, DC)
V.1-5, 1959-62. For publisher information, see JMCMAR.
Volume(issue)/page/year: 4,79,1961
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intraperitoneal
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 24500 ug/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
GCITA9 Gazzetta Chimica Italiana. (Societa Chimica Italiana, Rome, Italy)
V.1- 1871- Volume(issue)/page/year: 92,3,1962
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intravenous
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 11 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
JMPCAS Journal of Medicinal and Pharmaceutical Chemistry. (Washington, DC)
V.1-5, 1959-62. For publisher information, see JMCMAR.
Volume(issue)/page/year: 4,79,1961
*** END OF RECORD ***