*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : UX9648200
CHEMICAL NAME : 3-Pyrrolidinamine,
1-(10,11-dihydrodibenzo(b,f)thiepin-10-yl)-N-ethyl-,
dihydrochloride, hydrate, D-(R)-
LAST UPDATED : 198204
DATA ITEMS CITED : 1
MOLECULAR FORMULA : C20-H24-N2-S.2Cl-H.H2-O
MOLECULAR WEIGHT : 414.45
WISWESSER LINE NOTATION : T C676 BS&T&J I- AT5NTJ CM2 &GH 2 &QH
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* D-Dibenzo(b,f)thiepin, 10,11-dihydro-10-(3-ethylamino-1-pyrrolidinyl)-,
2HCl, hydrate
* 10-(D-(R)-3-Ethylaminopyrrolidino)-10,11-dihydrodibenzo(b,f)thiepin
dihydrochloride hydrate
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Intraperitoneal
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 160 mg/kg
TOXIC EFFECTS :
Behavioral - convulsions or effect on seizure threshold
Behavioral - changes in motor activity (specific assay)
Behavioral - ataxia
REFERENCE :
JMCMAR Journal of Medicinal Chemistry. (American Chemical Soc.,
Distribution Office Dept. 223, POB POB 57136, West End Stn., Washington, DC
20037) V.6- 1963- Volume(issue)/page/year: 17,690,1974
*** END OF RECORD ***