*** CHEMICAL IDENTIFICATION ***
RTECS NUMBER : UV7187000
CHEMICAL NAME : Pyrimidine, 5-bromo-2,4,6-tris(1-aziridinyl)-
CAS REGISTRY NUMBER : 13922-84-4
BEILSTEIN REFERENCE NO. : 0811811
REFERENCE : 5-25-12-00320 (Beilstein Handbook Reference)
LAST UPDATED : 199612
DATA ITEMS CITED : 2
MOLECULAR FORMULA : C10-H12-Br-N5
MOLECULAR WEIGHT : 282.18
WISWESSER LINE NOTATION : T6N CNJ B- AT3NTJ& D- AT3NTJ& EE F- AT3NTJ
COMPOUND DESCRIPTOR : Drug
SYNONYMS/TRADE NAMES :
* 5-Bromo-2,4,6-tris(1-aziridinyl)pyrimidine
* 2,4,6-Tri(ethyleneimino)-5-bromopyrimidine
*** HEALTH HAZARD DATA ***
** ACUTE TOXICITY DATA **
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Parenteral
SPECIES OBSERVED : Rodent - rat
DOSE/DURATION : 1150 ug/kg
TOXIC EFFECTS :
Behavioral - changes in motor activity (specific assay)
Behavioral - muscle contraction or spasticity
Lungs, Thorax, or Respiration - dyspnea
REFERENCE :
FATOBP Farmakologiya i Toksikologiya (Kiev). Pharmacology and Toxicology.
(Kievskii Nauchno- Issledovatel'skii Institut Farmakologii i Toksikologii,
Kiev, USSR) No.1- 1964- Volume(issue)/page/year: 5,101,1970
TYPE OF TEST : LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE : Parenteral
SPECIES OBSERVED : Rodent - mouse
DOSE/DURATION : 5500 ug/kg
TOXIC EFFECTS :
Behavioral - changes in motor activity (specific assay)
Behavioral - muscle contraction or spasticity
Lungs, Thorax, or Respiration - dyspnea
REFERENCE :
FATOBP Farmakologiya i Toksikologiya (Kiev). Pharmacology and Toxicology.
(Kievskii Nauchno- Issledovatel'skii Institut Farmakologii i Toksikologii,
Kiev, USSR) No.1- 1964- Volume(issue)/page/year: 5,101,1970
*** END OF RECORD ***